The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
28256371 |
83 |
Synthesis of bulky-tailed sulfonamides incorporating pyrido[2,3-d][1,2,4]triazolo[4,3-a]pyrimidin-1(5H)-yl) moieties and evaluation of their carbonic anhydrases I, II, IV and IX inhibitory effects. |
University of Wollongong |
28161252 |
64 |
Synthesis and biological evaluation of cyclic imides incorporating benzenesulfonamide moieties as carbonic anhydrase I, II, IV and IX inhibitors. |
King Saud University |
28237553 |
76 |
Human carbonic anhydrase inhibitory profile of mono- and bis-sulfonamides synthesized via a direct sulfochlorination of 3- and 4-(hetero)arylisoxazol-5-amine scaffolds. |
Saint Petersburg State University |
28109946 |
84 |
Novel indolin-2-one-based sulfonamides as carbonic anhydrase inhibitors: Synthesis, in vitro biological evaluation against carbonic anhydrases isoforms I, II, IV and VII and molecular docking studies. |
Kafrelsheikh University |
28075587 |
102 |
Design and Synthesis of Novel Nonsteroidal Anti-Inflammatory Drugs and Carbonic Anhydrase Inhibitors Hybrids (NSAIDs-CAIs) for the Treatment of Rheumatoid Arthritis. |
University of Florence |
12565948 |
120 |
Modelling of carbonic anhydrase inhibitory activity of sulfonamides using molecular negentropy. |
A.P.S. University |
28111158 |
100 |
Synthesis of isoxazole-containing sulfonamides with potent carbonic anhydrase II and VII inhibitory properties. |
Abant Izzet Baysal University |
27919611 |
60 |
Discovery of 4-sulfamoyl-phenyl-ß-lactams as a new class of potent carbonic anhydrase isoforms I, II, IV and VII inhibitors: The first example of subnanomolar CA IV inhibitors. |
National Institute of Pharmaceutical Education and Research (NIPER) |
27876475 |
68 |
Microwave assisted synthesis of novel tetrazole/sulfonamide derivatives based on octahydroacridine, xanthene and chromene skeletons as inhibitors of the carbonic anhydrases isoforms I, II, IV and VII. |
Dumlupinar University |
27144971 |
60 |
PEGylated Bis-Sulfonamide Carbonic Anhydrase Inhibitors Can Efficiently Control the Growth of Several Carbonic Anhydrase IX-Expressing Carcinomas. |
Temple University |
27172398 |
20 |
An Unusual Natural Product Primary Sulfonamide: Synthesis, Carbonic Anhydrase Inhibition, and Protein X-ray Structures of Psammaplin C. |
Griffith University |
27298005 |
92 |
Microwave assisted synthesis of novel acridine-acetazolamide conjugates and investigation of their inhibition effects on human carbonic anhydrase isoforms hCA I, II, IV and VII. |
Dumlupinar University |
26498394 |
105 |
Inhibition of mammalian carbonic anhydrase isoforms I-XIV with a series of phenolic acid esters. |
Universit£ |
26498393 |
116 |
New natural product carbonic anhydrase inhibitors incorporating phenol moieties. |
Aristotle University of Thessaloniki |
26347950 |
32 |
Phosphate Chemical Probes Designed for Location Specific Inhibition of Intracellular Carbonic Anhydrases. |
Griffith University |
25468040 |
77 |
Inhibition studies of new ureido-substituted sulfonamides incorporating a GABA moiety against human carbonic anhydrase isoforms I-XIV. |
TBA |
25358084 |
143 |
Discovery and characterization of novel selective inhibitors of carbonic anhydrase IX. |
Vilnius University |
24689792 |
54 |
Cyclic secondary sulfonamides: unusually good inhibitors of cancer-related carbonic anhydrase enzymes. |
Griffith University |
23010455 |
108 |
Synthesis of C-cinnamoyl glycosides and their inhibitory activity against mammalian carbonic anhydrases. |
Universidad Nacional De La Plata |
23067387 |
105 |
Tricyclic sulfonamides incorporating benzothiopyrano[4,3-c]pyrazole and pyridothiopyrano[4,3-c]pyrazole effectively inhibita- andß-carbonic anhydrase: X-ray crystallography and solution investigations on 15 isoforms. |
Universit£ |
22687439 |
51 |
Synthesis and carbonic anhydrase inhibitory properties of novel bromophenols and their derivatives including natural products: vidalol B. |
Atat£Rk University |
22487176 |
109 |
Flavones and structurally related 4-chromenones inhibit carbonic anhydrases by a different mechanism of action compared to coumarins. |
Universit£ |
21211980 |
47 |
Characterization and anions inhibition studies of ana-carbonic anhydrase from the teleost fish Dicentrarchus labrax. |
Ondokuz Mayis University |
20674354 |
79 |
Carbonic anhydrase inhibitors. Antioxidant polyphenols effectively inhibit mammalian isoforms I-XV. |
Universit£ |
20605094 |
91 |
Carbonic anhydrase inhibitors. The X-ray crystal structure of human isoform II in adduct with an adamantyl analogue of acetazolamide resides in a less utilized binding pocket than most hydrophobic inhibitors. |
University of Florida |
20472429 |
80 |
Carbonic anhydrase inhibitors: crystallographic and solution binding studies for the interaction of a boron-containing aromatic sulfamide with mammalian isoforms I-XV. |
Istituto Di Biostrutture E Bioimmagini-Cnr |
20363633 |
67 |
Thioether benzenesulfonamide inhibitors of carbonic anhydrases II and IV: structure-based drug design, synthesis, and biological evaluation. |
Pfizer |
20185318 |
132 |
Carbonic anhydrase inhibitors. Inhibition of mammalian isoforms I-XIV with a series of natural product polyphenols and phenolic acids. |
Universit£ |
19911821 |
273 |
Deciphering the mechanism of carbonic anhydrase inhibition with coumarins and thiocoumarins. |
Universita Degli Studi Di Firenze |
19854054 |
18 |
Nitric oxide-donating carbonic anhydrase inhibitors for the treatment of open-angle glaucoma. |
Nicox Research Institute |
20028100 |
78 |
The coumarin-binding site in carbonic anhydrase accommodates structurally diverse inhibitors: the antiepileptic lacosamide as an example and lead molecule for novel classes of carbonic anhydrase inhibitors. |
Universit£ |
19269822 |
75 |
Carbonic anhydrase inhibitors. Inhibition of cytosolic isoforms I, II, III, VII and XIII with less investigated inorganic anions. |
Universit£ |
19186056 |
60 |
A thiabendazole sulfonamide shows potent inhibitory activity against mammalian and nematode alpha-carbonic anhydrases. |
Universit£ |
18990571 |
65 |
Carbonic anhydrase inhibitors: 2-substituted-1,3,4-thiadiazole-5-sulfamides act as powerful and selective inhibitors of the mitochondrial isozymes VA and VB over the cytosolic and membrane-associated carbonic anhydrases I, II and IV. |
Ecole Nationale Sup£Rieure De Chimie De Montpellier |
18359629 |
84 |
Carbonic anhydrase inhibitors: the X-ray crystal structure of ethoxzolamide complexed to human isoform II reveals the importance of thr200 and gln92 for obtaining tight-binding inhibitors. |
Istituto Di Biostrutture E Bioimmagini-Cnr |
17475500 |
130 |
Carbonic anhydrases as targets for medicinal chemistry. |
Universit£ |
17376683 |
63 |
Carbonic anhydrase inhibitors. Inhibition of isoforms I, II, IV, VA, VII, IX, and XIV with sulfonamides incorporating fructopyranose-thioureido tails. |
Ecole Nationale Sup£Rieure De Chimie De Montpellier |
17314045 |
11 |
Phosph(on)ate as a zinc-binding group in metalloenzyme inhibitors: X-ray crystal structure of the antiviral drug foscarnet complexed to human carbonic anhydrase I. |
Universit£ |
16290146 |
30 |
Carbonic anhydrase inhibitors: Valdecoxib binds to a different active site region of the human isoform II as compared to the structurally related cyclooxygenase II"selective" inhibitor celecoxib. |
Istituto Di Biostrutture E Bioimmagini-Cnr |
15686931 |
84 |
Carbonic anhydrase inhibitors. Inhibition of the membrane-bound human and bovine isozymes IV with sulfonamides. |
Universit£ |
15664814 |
55 |
Carbonic anhydrase inhibitors. Inhibition of isozymes I, II, IV, V, and IX with anions isosteric and isoelectronic with sulfate, nitrate, and carbonate. |
Universit£ |
15501038 |
68 |
Carbonic anhydrase inhibitors: inhibition of the membrane-bound human isozyme IV with anions. |
Universit£ |
15357993 |
82 |
Carbonic anhydrase inhibitors. Inhibition of the beta-class enzyme from the methanoarchaeon Methanobacterium thermoautotrophicum (Cab) with anions. |
Universit£ |
15139757 |
105 |
Carbonic anhydrase inhibitors: synthesis and topical intraocular pressure lowering effects of fluorine-containing inhibitors devoid of enhanced reactivity. |
Universit£ |
11906288 |
713 |
Carbonic anhydrase inhibitors. A general approach for the preparation of water-soluble sulfonamides incorporating polyamino-polycarboxylate tails and of their metal complexes possessing long-lasting, topical intraocular pressure-lowering properties. |
Universit£ |
11784136 |
100 |
Carbonic anhydrase inhibitors: anticonvulsant sulfonamides incorporating valproyl and other lipophilic moieties. |
University of Namur |
11123998 |
141 |
Carbonic anhydrase inhibitors: water-soluble 4-sulfamoylphenylthioureas as topical intraocular pressure-lowering agents with long-lasting effects. |
Universit£ |
11087579 |
465 |
Carbonic anhydrase inhibitors: perfluoroalkyl/aryl-substituted derivatives of aromatic/heterocyclic sulfonamides as topical intraocular pressure-lowering agents with prolonged duration of action. |
Universit£ |
10479300 |
383 |
Carbonic anhydrase inhibitors: synthesis of water-soluble, aminoacyl/dipeptidyl sulfonamides possessing long-lasting intraocular pressure-lowering properties via the topical route. |
Universit£ |
10411484 |
176 |
Carbonic anhydrase inhibitors. Synthesis of water-soluble, topically effective, intraocular pressure-lowering aromatic/heterocyclic sulfonamides containing cationic or anionic moieties: is the tail more important than the ring? |
Universit£ |
15012984 |
192 |
Carbonic anhydrase inhibitors: the first selective, membrane-impermeant inhibitors targeting the tumor-associated isozyme IX. |
Slovak Academy of Sciences |
14698154 |
26 |
Carbonic anhydrase inhibitors: X-ray crystallographic structure of the adduct of human isozyme II with the antipsychotic drug sulpiride. |
Bruker-Axs |
14684331 |
24 |
Carbonic anhydrase inhibitors: E7070, a sulfonamide anticancer agent, potently inhibits cytosolic isozymes I and II, and transmembrane, tumor-associated isozyme IX. |
Universit£ |
12643899 |
127 |
Carbonic anhydrase inhibitors: inhibition of the tumor-associated isozyme IX with aromatic and heterocyclic sulfonamides. |
Universit£ |
12617904 |
46 |
Carbonic anhydrase inhibitors: SAR and X-ray crystallographic study for the interaction of sugar sulfamates/sulfamides with isozymes I, II and IV. |
Universit£ |
14611846 |
101 |
Carbonic anhydrase inhibitors: topically acting antiglaucoma sulfonamides incorporating esters and amides of 3- and 4-carboxybenzolamide. |
Universit£ |
12039560 |
377 |
Carbonic anhydrase inhibitors. Preparation of potent sulfonamides inhibitors incorporating bile acid tails. |
Universit£ |
11229775 |
204 |
Carbonic anhydrase inhibitors: synthesis of sulfonamides incorporating dtpa tails and of their zinc complexes with powerful topical antiglaucoma properties. |
Universit£ |
11425561 |
197 |
Carbonic anhydrase inhibitors: 4-sulfamoyl-benzenecarboxamides and 4-chloro-3-sulfamoyl-benzenecarboxamides with strong topical antiglaucoma properties. |
Universit£ |
10762051 |
66 |
Carbonic anhydrase inhibitors: topical sulfonamide antiglaucoma agents incorporating secondary amine moieties. |
Universit£ |
10843231 |
129 |
Carbonic anhydrase inhibitors: synthesis of N-morpholylthiocarbonylsulfenylamino aromatic/heterocyclic sulfonamides and their interaction with isozymes I, II and IV. |
Universit£ |
22365761 |
144 |
New chemotypes acting as isozyme-selective carbonic anhydrase inhibitors with low affinity for the offtarget cytosolic isoform II. |
Universit£ |
22245047 |
135 |
Structure-activity relationships for the interaction of 5,10-dihydroindeno[1,2-b]indole derivatives with human and bovine carbonic anhydrase isoforms I, II, III, IV and VI. |
Ondokuz Mayis University |
22230050 |
82 |
Synthesis and carbonic anhydrase inhibitory properties of novel cyclohexanonyl bromophenol derivatives. |
Artvin£Oruh University |
21821413 |
65 |
Synthesis of rhodamine B-benzenesulfonamide conjugates and their inhibitory activity against humana- and bacterial/fungalß-carbonic anhydrases. |
Ecole Nationale Sup£Rieure De Chimie De Montpellier |
21515057 |
153 |
Sulfonamides incorporating 1,3,5-triazine moieties selectively and potently inhibit carbonic anhydrase transmembrane isoforms IX, XII and XIV over cytosolic isoforms I and II: Solution and X-ray crystallographic studies. |
Universit£ |
21549597 |
71 |
Synthesis and crystallographic analysis of new sulfonamides incorporating NO-donating moieties with potent antiglaucoma action. |
U.O. Oculistica Az. Usl 3 |
21377369 |
60 |
Purification and inhibition studies with anions and sulfonamides of ana-carbonic anhydrase from the Antarctic seal Leptonychotes weddellii. |
Universit£ |
20590092 |
273 |
Polyamines inhibit carbonic anhydrases by anchoring to the zinc-coordinated water molecule. |
Universita Degli Studi Di Firenze |
19527930 |
53 |
The protein tyrosine kinase inhibitors imatinib and nilotinib strongly inhibit several mammalian alpha-carbonic anhydrase isoforms. |
University of Tampere and Tampere University Hospital |
19121582 |
15 |
Carbonic anhydrase inhibitors: inhibition studies of a coral secretory isoform with inorganic anions. |
Centre Scientifique De Monaco |
16759856 |
9 |
N-hydroxyurea--a versatile zinc binding function in the design of metalloenzyme inhibitors. |
Università |
15780631 |
55 |
Carbonic anhydrase inhibitors. Inhibition of isozymes I, II, IV, V and IX with complex fluorides, chlorides and cyanides. |
Università |
15745821 |
21 |
Carbonic anhydrase inhibitors. Interaction of isozymes I, II, IV, V, and IX with organic phosphates and phosphonates. |
University of Montpellier |
15664815 |
45 |
Carbonic anhydrase inhibitors. Interaction of isozymes I, II, IV, V, and IX with carboxylates. |
Università |
15501037 |
27 |
Carbonic anhydrase inhibitors. Interaction of isozymes I, II, IV, V, and IX with phosphates, carbamoyl phosphate, and the phosphonate antiviral drug foscarnet. |
Università |
15081040 |
4 |
Carbonic anhydrase inhibitors: X-ray crystallographic structure of the adduct of human isozyme II with a topically acting antiglaucoma sulfonamide. |
Bruker-Axs |
12873509 |
4 |
Carbonic anhydrase inhibitors: X-ray crystallographic structure of the adduct of human isozyme II with a bis-sulfonamide-two heads are better than one? |
Università |
32519851 |
164 |
Sulfonamide Inhibitors of Human Carbonic Anhydrases Designed through a Three-Tails Approach: Improving Ligand/Isoform Matching and Selectivity of Action. |
University of Firenze |
32435377 |
30 |
Glycomimetic Based Approach toward Selective Carbonic Anhydrase Inhibitors. |
Universit£ |
30996772 |
55 |
-Nitrosulfonamides as Carbonic Anhydrase Inhibitors: A Promising Chemotype for Targeting Chagas Disease and Leishmaniasis. |
University of Florence |
10649985 |
390 |
Carbonic anhydrase inhibitors: synthesis of membrane-impermeant low molecular weight sulfonamides possessing in vivo selectivity for the membrane-bound versus cytosolic isozymes. |
Università |
32364386 |
184 |
Phenyl(thio)phosphon(amid)ate Benzenesulfonamides as Potent and Selective Inhibitors of Human Carbonic Anhydrases II and VII Counteract Allodynia in a Mouse Model of Oxaliplatin-Induced Neuropathy. |
University of Florence |
32031797 |
96 |
Discovery of Potent Dual-Tailed Benzenesulfonamide Inhibitors of Human Carbonic Anhydrases Implicated in Glaucoma and in Vivo Profiling of Their Intraocular Pressure-Lowering Action. |
University of Wollongong |
31255926 |
46 |
Sulfamates in drug design and discovery: Pre-clinical and clinical investigations. |
University of Sharjah |
31794211 |
138 |
"A Sweet Combination": Developing Saccharin and Acesulfame K Structures for Selectively Targeting the Tumor-Associated Carbonic Anhydrases IX and XII. |
University of Florence |
31515057 |
20 |
Highly hydrophilic 1,3-oxazol-5-yl benzenesulfonamide inhibitors of carbonic anhydrase II for reduction of glaucoma-related intraocular pressure. |
Saint Petersburg State University |
31476557 |
164 |
From random to rational: A discovery approach to selective subnanomolar inhibitors of human carbonic anhydrase IV based on the Castagnoli-Cushman multicomponent reaction. |
Saint Petersburg State University |
31401537 |
45 |
Synthesis of novel tellurides bearing benzensulfonamide moiety as carbonic anhydrase inhibitors with antitumor activity. |
University of Florence |
31287314 |
52 |
Synthesis and Evaluation of Carbonic Anhydrase Inhibitors with Carbon Monoxide Releasing Properties for the Management of Rheumatoid Arthritis. |
Universit£ |
31136893 |
176 |
Benzensulfonamides bearing spyrohydantoin moieties act as potent inhibitors of human carbonic anhydrases II and VII and show neuropathic pain attenuating effects. |
University of Florence |
31740053 |
1887 |
Halogenated and di-substituted benzenesulfonamides as selective inhibitors of carbonic anhydrase isoforms. |
Vilnius University |
31539777 |
92 |
Continued exploration and tail approach synthesis of benzenesulfonamides containing triazole and dual triazole moieties as carbonic anhydrase I, II, IV and IX inhibitors. |
Kurukshetra University |
30553625 |
761 |
Pyrrolidinone-bearing methylated and halogenated benzenesulfonamides as inhibitors of carbonic anhydrases. |
Kaunas University of Technology |
31413806 |
65 |
Bis-benzoxaboroles: Design, Synthesis, and Biological Evaluation as Carbonic Anhydrase Inhibitors. |
Universit£ |
26678172 |
70 |
Inhibition of carbonic anhydrase isoforms I, II, IV, VII and XII with carboxylates and sulfonamides incorporating phthalimide/phthalic anhydride scaffolds. |
King Saud University |
24300919 |
55 |
Combining the tail and the ring approaches for obtaining potent and isoform-selective carbonic anhydrase inhibitors: solution and X-ray crystallographic studies. |
Universit£ |
24103430 |
78 |
Inhibition of human carbonic anhydrase isoforms I-XIV with sulfonamides incorporating fluorine and 1,3,5-triazine moieties. |
Universit£ |
30496988 |
25 |
Pharmaceutical and medicinal significance of sulfur (S |
Wuhan University of Technology |
16458003 |
158 |
QSAR study on topically acting sulfonamides incorporating GABA moieties: a molecular connectivity approach. |
A.P.S. University |
11831900 |
8 |
Structural aspects of isozyme selectivity in the binding of inhibitors to carbonic anhydrases II and IV. |
University of Pennsylvania |
30193219 |
114 |
Discovery of new 2, 5-disubstituted 1,3-selenazoles as selective human carbonic anhydrase IX inhibitors with potent anti-tumor activity. |
Department of University of Florence |
30344913 |
24 |
Famotidine, an Antiulcer Agent, Strongly Inhibits |
University of Florence |
29685656 |
8 |
Synthesis, structure and bioactivity of primary sulfamate-containing natural products. |
Griffith University |
29571155 |
124 |
Synthesis of novel 4-functionalized 1,5-diaryl-1,2,3-triazoles containing benzenesulfonamide moiety as carbonic anhydrase I, II, IV and IX inhibitors. |
Kurukshetra University |
28947945 |
72 |
Discovery of New Selenoureido Analogues of 4-(4-Fluorophenylureido)benzenesulfonamide as Carbonic Anhydrase Inhibitors. |
University of Florence |
28802125 |
92 |
Novel 4/3-((4-oxo-5-(2-oxoindolin-3-ylidene)thiazolidin-2-ylidene)amino) benzenesulfonamides: Synthesis, carbonic anhydrase inhibitory activity, anticancer activity and molecular modelling studies. |
Kafrelsheikh University |
29746127 |
195 |
Discovery of Novel Nonsteroidal Anti-Inflammatory Drugs and Carbonic Anhydrase Inhibitors Hybrids (NSAIDs-CAIs) for the Management of Rheumatoid Arthritis. |
Ege University Bornova |
29305297 |
480 |
Benzimidazole design, synthesis, and docking to build selective carbonic anhydrase VA inhibitors. |
Vilnius University |
30006175 |
644 |
Design of two-tail compounds with rotationally fixed benzenesulfonamide ring as inhibitors of carbonic anhydrases. |
Vilnius University |
29909339 |
84 |
Design and synthesis of novel benzenesulfonamide containing 1,2,3-triazoles as potent human carbonic anhydrase isoforms I, II, IV and IX inhibitors. |
Kurukshetra University |
29684705 |
72 |
Dual-tail arylsulfone-based benzenesulfonamides differently match the hydrophobic and hydrophilic halves of human carbonic anhydrases active sites: Selective inhibitors for the tumor-associated hCA IX isoform. |
Egyptian Russian University |
29635168 |
140 |
2-Benzylpiperazine: A new scaffold for potent human carbonic anhydrase inhibitors. Synthesis, enzyme inhibition, enantioselectivity, computational and crystallographic studies and in vivo activity for a new class of intraocular pressure lowering agents. |
University of Florence |
29912561 |
40 |
4-Substituted Benzenesulfonamides Incorporating Bi/Tricyclic Moieties Act as Potent and Isoform-Selective Carbonic Anhydrase II/IX Inhibitors. |
Universit£ |
29259736 |
70 |
Synthesis of Novel Selenides Bearing Benzenesulfonamide Moieties as Carbonic Anhydrase I, II, IV, VII, and IX Inhibitors. |
University of Florence |
29259754 |
76 |
Discovery of New Sulfonamide Carbonic Anhydrase IX Inhibitors Incorporating Nitrogenous Bases. |
University of Florence |
29057059 |
82 |
Lucky Switcheroo: Dramatic Potency and Selectivity Improvement of Imidazoline Inhibitors of Human Carbonic Anhydrase VII. |
Saint Petersburg State University |
28277280 |
43 |
Bortezomib inhibits mammalian carbonic anhydrases. |
Universit£ |
28302505 |
120 |
Evaluation of selenide, diselenide and selenoheterocycle derivatives as carbonic anhydrase I, II, IV, VII and IX inhibitors. |
Universit£ |
23914927 |
24 |
Inhibition of mammalian carbonic anhydrases I-XIV with grayanotoxin III: solution and in silico studies. |
University of Calgary |
22299585 |
46 |
Analysis of saponins and phenolic compounds as inhibitors of a-carbonic anhydrase isoenzymes. |
Ege University |
22299576 |
44 |
Metronidazole-coumarin conjugates and 3-cyano-7-hydroxy-coumarin act as isoform-selective carbonic anhydrase inhibitors. |
Ecole Nationale Superieure De Chimie De Montpellier |
22299577 |
12 |
Three new aromatic sulfonamide inhibitors of carbonic anhydrases I, II, IV and XII. |
Universit?? Di Firenze |
22168126 |
43 |
Carbonic anhydrase inhibitors: in vitro inhibition of a isoforms (hCA I, hCA II, bCA III, hCA IV) by flavonoids. |
Ondokuz Mayis University |
22145694 |
64 |
Simple methanesulfonates are hydrolyzed by the sulfatase carbonic anhydrase activity. |
Agri Ibrahim Cecen University |
22050606 |
36 |
a-Carbonic anhydrases are sulfatases with cyclic diol monosulfate esters. |
Dumlupinar University |
15499999 |
35 |
Benzolamide is not a membrane-impermeant carbonic anhydrase inhibitor. |
UniversitÀ Degli Studi Di Firenze |
11916140 |
21 |
Carbonic anhydrase activity modulators: synthesis of inhibitors and activators incorporating 2-substituted-thiazol-4-yl-methyl scaffolds. |
UniversitÀ |
19703035 |
60 |
Which carbonic anhydrases are targeted by the antiepileptic sulfonamides and sulfamates? |
Istituto Di Biostrutture E Bioimmagini-Cnr |
19731956 |
72 |
Carbonic anhydrase inhibitors. Comparison of aliphatic sulfamate/bis-sulfamate adducts with isozymes II and IX as a platform for designing tight-binding, more isoform-selective inhibitors. |
Cnr |
19119014 |
12 |
Carbonic anhydrase inhibitors. Comparison of chlorthalidone, indapamide, trichloromethiazide, and furosemide X-ray crystal structures in adducts with isozyme II, when several water molecules make the difference. |
Universita Degli Studi Di Firenze |
19128966 |
80 |
Carbonic anhydrase inhibitors: the membrane-associated isoform XV is highly inhibited by inorganic anions. |
Universita Degli Studi Di Firenze |
18579385 |
132 |
Carbonic anhydrase inhibitors: inhibition of mammalian isoforms I-XIV with a series of substituted phenols including paracetamol and salicylic acid. |
Universita Degli Studi Di Firenze |
18819811 |
195 |
Carbonic anhydrase inhibitors: synthesis and inhibition studies against mammalian isoforms I-XV with a series of 2-(hydrazinocarbonyl)-3-substituted-phenyl-1H-indole-5-sulfonamides. |
Istanbul University |
18374572 |
100 |
Carbonic anhydrase inhibitors. Interaction of indapamide and related diuretics with 12 mammalian isozymes and X-ray crystallographic studies for the indapamide-isozyme II adduct. |
Universita Degli Studi Di Firenze |
18640037 |
48 |
Carbonic anhydrase inhibitors. Interaction of the antitumor sulfamate EMD 486019 with twelve mammalian carbonic anhydrase isoforms: Kinetic and X-ray crystallographic studies. |
Universita Degli Studi Di Firenze |
14971907 |
180 |
Carbonic anhydrase inhibitors. Inhibition of mitochondrial isozyme V with aromatic and heterocyclic sulfonamides. |
Universita Degli Studi Di Firenze |
15084132 |
88 |
Carbonic anhydrase inhibitors. Design of selective, membrane-impermeant inhibitors targeting the human tumor-associated isozyme IX. |
Canadian Institutes of Health Research |
14736236 |
20 |
Unexpected nanomolar inhibition of carbonic anhydrase by COX-2-selective celecoxib: new pharmacological opportunities due to related binding site recognition. |
University of Marburg |
17125255 |
77 |
Carbonic anhydrase inhibitors: clash with Ala65 as a means for designing inhibitors with low affinity for the ubiquitous isozyme II, exemplified by the crystal structure of the topiramate sulfamide analogue. |
Universite Montpellier Ii |
12747790 |
171 |
Carbonic anhydrase inhibitors. Inhibition of tumor-associated isozyme IX by halogenosulfanilamide and halogenophenylaminobenzolamide derivatives. |
University of Agricultural Sciences and Veterinary Medicine |
10882008 |
93 |
2H-Thieno[3,2-e]- and [2,3-e]-1,2-thiazine-6-sulfonamide 1,1-dioxides as ocular hypotensive agents: synthesis, carbonic anhydrase inhibition and evaluation in the rabbit. |
Alcon Research |
11020282 |
512 |
Carbonic anhydrase and matrix metalloproteinase inhibitors: sulfonylated amino acid hydroxamates with MMP inhibitory properties act as efficient inhibitors of CA isozymes I, II, and IV, and N-hydroxysulfonamides inhibit both these zinc enzymes. |
Universita Degli Studi |